Xanomeline tartrate

CAS No. 152854-19-8

Xanomeline tartrate( —— )

Catalog No. M35083 CAS No. 152854-19-8

Xanomeline tartrate (LY 246708 tartrate) is an M1 and M4 mAChR agonist with antipsychotic-like activity that improves cognition and can be used in studies of schizophrenia and Alzheimer's disease.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 44 In Stock
10MG 61 In Stock
25MG 90 In Stock
50MG 136 In Stock
100MG 195 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Xanomeline tartrate
  • Note
    Research use only, not for human use.
  • Brief Description
    Xanomeline tartrate (LY 246708 tartrate) is an M1 and M4 mAChR agonist with antipsychotic-like activity that improves cognition and can be used in studies of schizophrenia and Alzheimer's disease.
  • Description
    Xanomeline (LY 246708) is the potent agonist of muscarinic M1/M4 receptor with antipsychotic-like activity. Xanomeline (LY 246708) increases neuronal excitability.Xanomeline (LY 246708) can be used for the research of schizophrenia.
  • In Vitro
    ——
  • In Vivo
    Animal Model:Male Cebus apella monkeys Dosage:0.5-3 mg/kg Administration:s.c.; 1-3 hours Result:Induced salivation and vomiting in some monkeys.
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    Others
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    152854-19-8
  • Formula Weight
    431.5
  • Molecular Formula
    C18H29N3O7S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 250 mg/mL (579.37 mM; Ultrasonic )
  • SMILES
    O[C@@H]([C@H](O)C(O)=O)C(O)=O.CCCCCCOc1nsnc1C1=CCCN(C)C1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Kreir M, et al. Role of Kv7.2/Kv7.3 and M1 muscarinic receptors in the regulation of neuronal excitability in hiPSC-derived neurons. Eur J Pharmacol. 2019;858:172474. ?
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